SCHEMBL13136348

SCHEMBL13136348

COC(=O)COCc1ncc(-c2cccc(Nc3cc(C)ccn3)n2)s1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SYK P43405 9/20 0.51
KARS1 Q15046 9/20 0.48
KDR P35968 1/20 0.41
JAK2 O60674 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2869572 0.92 SYK (0.53) SYKKARS1KDRJAK2
SCHEMBL13136341 0.91 SYK (0.51) SYKKARS1KDRJAK2
Hydrochloric Acid SCHEMBL2868657 0.91 SYK (0.53) SYKKARS1KDRJAK2
SCHEMBL13136354 0.90 SYK (0.50) SYKKARS1KDRJAK2
SCHEMBL13136355 0.89 SYK (0.49) SYKKARS1KDR
SCHEMBL13136166 0.85 SYK (0.51) SYKKARS1KDR
SCHEMBL13136359 0.85 SYK (0.51) SYKKARS1
SCHEMBL13136069 0.84 SYK (0.50) SYKKARS1KDR
SCHEMBL13136356 0.84 SYK (0.49) SYKKARS1
SCHEMBL13136195 0.84 SYK (0.49) SYKKARS1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7803801-B2 Aminopyridine compounds having Syk inhibitory activity JAPAN TOBACCO, INC. (JP) 2010-09-28 US disclosed
US-7803801-B2 Aminopyridine compounds having Syk inhibitory activity JAPAN TOBACCO, INC. (JP) 2010-09-28 US disclosed