SCHEMBL1315

SCHEMBL1315

Cc1c(CO[Si](C)(C)C)ncn1S(=O)(=O)N(C)C

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL713 0.78 KDM4E (0.46) KDM4EGAATSHRSMN1; SMN2
SCHEMBL993 0.78 KDM4E (0.46) KDM4EGAATSHRSMN1; SMN2
SCHEMBL22075818 0.72 KDM4E (0.53) KDM4EGAATSHRSMN1; SMN2
SCHEMBL7267947 0.67 KDM4E (0.47) KDM4EGAATSHRSMN1; SMN2
SCHEMBL9876336 0.64 TSHR (0.42) KDM4EGAATSHRSMN1; SMN2
SCHEMBL1056 0.62 KDM4E (0.39) KDM4EGAATSHR
SCHEMBL941 0.62 TSHR (0.40) KDM4EGAATSHRSMN1; SMN2
SCHEMBL14334526 0.59 FGFR1 (0.40) KDM4EGAATSHRSMN1; SMN2
SCHEMBL31460301 0.59 GAA (1.00) KDM4EGAATSHRSMN1; SMN2
SCHEMBL16125139 0.59 KDM4E (0.31) KDM4EGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360800-A Tetrahydro-1H-pyrido[4,3-b]indol-1-one derivatives GLAXO GROUP LIMITED (GB) 1994-11-01 US disclosed
EP-0306323-A2 Lactam derivatives GLAXO GROUP LIMITED (GB) 1989-03-08 EP disclosed