SCHEMBL13153809

SCHEMBL13153809

O=c1c2nn(Cc3ccc(N4CCC=N4)cc3)c3ccsc3c-2nn1C1CCCOC1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.32
PDE4A P27815 2/20 0.32
PDE4B Q07343 2/20 0.32
PDE4C Q08493 2/20 0.32
PDE4D Q08499 2/20 0.32
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL617769 0.86 FEN1 (0.36) FEN1PDE4APDE4BPDE4CPDE4D
SCHEMBL7911711 0.85 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL615989 0.82 CHRM1 (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL617714 0.79 PDE1B (0.35) FEN1PDE4APDE4BPDE4CPDE4D
SCHEMBL616912 0.78 FEN1 (0.35) FEN1PDE4APDE4BPDE4CPDE4D
SCHEMBL7910180 0.70 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7908279 0.70 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL3787499 0.69 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL3807036 0.68 CHRM1 (0.48) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL7906425 0.68 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010123716-A1 HETEROCYCLIC FUSED CINNOLINE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK SHARP & DOHME CORP. (US) 2010-10-28 WO disclosed