SCHEMBL13174703

SCHEMBL13174703

CC(C)(O)CC1CCN(C(=O)c2cc3ccc(Br)cc3[nH]2)CC1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 9/20 0.74
HRH4 Q9H3N8 2/20 0.63
GRIN2D O15399 3/20 0.53
GRIN3B O60391 3/20 0.53
GRIN1 Q05586 3/20 0.53
GRIN2A Q12879 3/20 0.53
GRIN2B Q13224 3/20 0.53
GRIN2C Q14957 3/20 0.53
GRIN3A Q8TCU5 3/20 0.53
HRH3 Q9Y5N1 1/20 0.51
MEN1 O00255 1/20 0.51
NPC1 O15118 1/20 0.51
KMT2A Q03164 1/20 0.51
GPR183 P32249 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3089444 0.91 AKR1C3 (0.78) AKR1C3HRH4GRIN2DGRIN3BGRIN1
SCHEMBL11981622 0.88 AKR1C3 (0.84) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL13174666 0.87 AKR1C3 (0.74) AKR1C3HRH4GRIN2DGRIN3BGRIN1
SCHEMBL13174668 0.87 AKR1C3 (0.74) AKR1C3HRH4GRIN2DGRIN3BGRIN1
SCHEMBL3101848 0.85 AKR1C3 (1.00) AKR1C3HRH4GRIN2DGRIN3BGRIN1
SCHEMBL3099610 0.85 AKR1C3 (0.85) AKR1C3HRH4GRIN2DGRIN3BGRIN1
SCHEMBL13173599 0.83 AKR1C3 (0.69) AKR1C3HRH4GRIN2DGRIN3BGRIN1
SCHEMBL3106410 0.83 AKR1C3 (0.72) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL13174677 0.82 AKR1C3 (0.71) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL13174701 0.82 AKR1C3 (0.71) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010101127-A1 INDOLE COMPOUND アステラス製薬株式会社 (JP) 2010-09-10 WO disclosed