SCHEMBL13186783

SCHEMBL13186783

COc1cccc2c1c(NS(=O)(=O)c1ccc(Cl)s1)nn2Cc1cccc(CNC(=O)C2CCCN2C)c1

nearest known ligand 0.82

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 20/20 0.82
CCR5 P51681 1/20 0.71
FFAR4 Q5NUL3 1/20 0.71
SLCO1B1 Q9Y6L6 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10235071 1.00 CCR4 (0.82) CCR4CCR5FFAR4SLCO1B1
SCHEMBL10235077 1.00 CCR4 (0.82) CCR4CCR5FFAR4SLCO1B1
SCHEMBL10235079 0.98 CCR4 (0.81) CCR4CCR5FFAR4SLCO1B1
Trifluoroacetic Acid SCHEMBL356776 0.96 CCR4 (0.76) CCR4CCR5FFAR4SLCO1B1
Trifluoroacetic Acid SCHEMBL358457 0.96 CCR4 (0.76) CCR4CCR5FFAR4SLCO1B1
Trifluoroacetic Acid SCHEMBL356159 0.94 CCR4 (0.75) CCR4CCR5FFAR4SLCO1B1
SCHEMBL356133 0.90 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1
SCHEMBL357175 0.89 CCR4 (0.70) CCR4CCR5FFAR4SLCO1B1
SCHEMBL357279 0.89 CCR4 (0.70) CCR4CCR5FFAR4SLCO1B1
Bicarbonate SCHEMBL15310366 0.88 CCR4 (0.86) CCR4CCR5FFAR4SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097395-A1 PYRAZOLE DERIVATIVES USED AS CCR4 RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-09-02 WO disclosed