SCHEMBL13186830

SCHEMBL13186830

COc1cccc2c1c(NS(=O)(=O)c1ccc(C)s1)nn2Cc1ccc(CNC(=O)C2COCCN2)cc1

nearest known ligand 0.80

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 20/20 0.80
CCR5 P51681 1/20 0.53
FFAR4 Q5NUL3 1/20 0.53
SLCO1B1 Q9Y6L6 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10279005 1.00 CCR4 (0.80) CCR4CCR5FFAR4SLCO1B1
Trifluoroacetic Acid SCHEMBL358432 0.96 CCR4 (0.74) CCR4CCR5FFAR4SLCO1B1
SCHEMBL10278781 0.95 CCR4 (0.87) CCR4CCR5FFAR4SLCO1B1
SCHEMBL13241520 0.95 CCR4 (0.87) CCR4CCR5FFAR4SLCO1B1
SCHEMBL13186841 0.95 CCR4 (0.87) CCR4CCR5FFAR4SLCO1B1
SCHEMBL10235306 0.93 CCR4 (0.91) CCR4CCR5FFAR4SLCO1B1
Trifluoroacetic Acid SCHEMBL357570 0.89 CCR4 (0.84) CCR4CCR5FFAR4SLCO1B1
SCHEMBL10234920 0.89 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1
SCHEMBL356525 0.89 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1
SCHEMBL10234917 0.89 CCR4 (1.00) CCR4CCR5FFAR4SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097395-A1 PYRAZOLE DERIVATIVES USED AS CCR4 RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2010-09-02 WO disclosed