SCHEMBL13234699

SCHEMBL13234699

CC(C)(C)c1cc(NC(=O)Nc2ccc(NC(=O)c3cc(Cl)cc(Cl)c3)cc2)no1

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 14/20 0.74
MAPK14 Q16539 1/20 0.66
CSF1R P07333 4/20 0.65
MEN1 O00255 1/20 0.65
NPC1 O15118 1/20 0.65
RAB9A P51151 1/20 0.65
KMT2A Q03164 1/20 0.65
RET P07949 2/20 0.62
PDGFRB P09619 2/20 0.62
KIT P10721 2/20 0.62
PDGFRA P16234 2/20 0.62
RAF1 P04049 4/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13234840 0.91 FLT3 (0.80) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234696 0.91 FLT3 (0.80) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234811 0.89 FLT3 (0.73) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234430 0.87 MAPK14 (0.76) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234704 0.85 FLT3 (1.00) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234760 0.84 FLT3 (0.82) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234771 0.84 FLT3 (0.82) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234373 0.84 FLT3 (1.00) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234769 0.84 FLT3 (1.00) FLT3MAPK14CSF1RMEN1NPC1
SCHEMBL13234806 0.84 FLT3 (0.71) FLT3MAPK14CSF1RMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100173917-A1 UREA DERIVATIVES AS ABL MODULATORS AMBIT BIOSCIENCES CORPORATION 2010-07-08 US disclosed
US-20100173917-A1 UREA DERIVATIVES AS ABL MODULATORS AMBIT BIOSCIENCES CORPORATION 2010-07-08 US disclosed
US-7750160-B2 Isoxazolyl urea derivatives as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-07-06 US disclosed
US-7750160-B2 Isoxazolyl urea derivatives as kinase modulators AMBIT BIOSCIENCES CORPORATION (US) 2010-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100173917-A1 UREA DERIVATIVES AS ABL MODULATORS ABL1, ABL2, BCR FLT3 7/4885MAPK14 1436/4885CSF1R 1746/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.