SCHEMBL13244249

SCHEMBL13244249

COc1nc(Cl)c2c(n1)NC(=O)C2

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.41
CYP1A2 P05177 1/20 0.34
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
CCNB2 O95067 1/20 0.31
CDK1 P06493 1/20 0.31
CCNB1 P14635 1/20 0.31
CCNB3 Q8WWL7 1/20 0.31
CMA1 P23946 1/20 0.31
AHR P35869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17926499 0.77 SRC (0.43) SRCCCNB2CDK1CCNB1CCNB3
SCHEMBL12019998 0.69 CYP1A2 (0.36) CYP1A2
SCHEMBL29319840 0.67 SRC (0.53) SRCCMA1AHR
SCHEMBL13244248 0.66 CYP1A2 (0.37) CYP1A2
SCHEMBL260293 0.65 TNNI3K (0.39) SRCCCNB2CDK1CCNB1CCNB3
SCHEMBL2821501 0.64
SCHEMBL13424558 0.62 MEN1 (0.42) SRCMEN1MAPTKMT2A
SCHEMBL2453854 0.62 SRC (0.56) SRCCMA1AHR
SCHEMBL2115445 0.62 CYP1A2 (0.68) CYP1A2MEN1ALDH1A1MAPTKMT2A
SCHEMBL275910 0.60 CYP1A2 (0.48) CYP1A2MEN1ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8338422-B2 Indolin-2-ones and aza-indolin-2-ones JANSSEN PHARMACEUTICA NV (BE) 2012-12-25 US disclosed
US-8338422-B2 Indolin-2-ones and aza-indolin-2-ones JANSSEN PHARMACEUTICA NV (BE) 2012-12-25 US disclosed
US-20100190786-A1 INDOLIN-2-ONES AND AZA-INDOLIN-2-ONES JANSSEN PHARMACEUTICA NV (BE) 2010-07-29 US disclosed
US-20100190786-A1 INDOLIN-2-ONES AND AZA-INDOLIN-2-ONES JANSSEN PHARMACEUTICA NV (BE) 2010-07-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100190786-A1 INDOLIN-2-ONES AND AZA-INDOLIN-2-ONES IDO2, IDO1, MKI67 SRC 1560/4885CYP1A2 1065/4885MEN1 1712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.