SCHEMBL13253299

SCHEMBL13253299

Cc1ccc(OC(C)(C)C(=O)N[C@@H](C)[C@@H](Cc2ccc(OCC[18F])cc2)c2cccc(C#N)c2)nc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 20/20 1.00
CNR2 P34972 6/20 1.00
CYP2D6 P10635 1/20 0.68
CYP2C9 P11712 1/20 0.68
KCNH2 Q12809 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3476142 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL30510967 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3476144 1.00 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3476704 0.94 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3476702 0.94 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3477587 0.93 CNR1 (0.89) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3477591 0.93 CNR1 (0.89) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3474186 0.92 CNR1 (0.87) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL13253309 0.92 CNR1 (1.00) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3476532 0.92 CNR1 (0.84) CNR1CNR2CYP2D6CYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7754188-B2 Radiolabeled cannabinoid-1 receptor modulators MERCK SHARP & DOHME CORP. (US) 2010-07-13 US disclosed