SCHEMBL13256367

SCHEMBL13256367

Cc1cc(C2CC2)ccc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.43
POLQ O75417 1/20 0.41
KDM1A O60341 1/20 0.39
HTR2C P28335 4/20 0.38
PDK2 Q15119 1/20 0.37
ESR2 Q92731 1/20 0.37
NOTUM Q6P988 2/20 0.37
PDE2A O00408 1/20 0.37
DRD2 P14416 1/20 0.35
DAO P14920 1/20 0.34
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13256370 0.93 HTR2A (0.48) HTR2APOLQKDM1AHTR2CPDK2
SCHEMBL30228395 0.88 HTR2C (0.56) HTR2AHTR2C
Hydrochloric Acid SCHEMBL4890973 0.87 HTR2C (0.57) HTR2AHTR2C
SCHEMBL18162314 0.85 POLQ (0.47) HTR2APOLQKDM1AHTR2CPDK2
SCHEMBL3434595 0.85 POLQ (0.47) HTR2APOLQKDM1AHTR2CPDK2
SCHEMBL18162311 0.84 POLQ (0.44) HTR2APOLQHTR2CPDK2NOTUM
SCHEMBL26020142 0.82 SSTR4 (0.35) HTR2AHTR2CPDK2ESR2PDE2A
SCHEMBL26020163 0.79 POLQ (0.43) HTR2APOLQKDM1AHTR2CPDK2
SCHEMBL13002296 0.79 KDM1A (0.53) HTR2APOLQKDM1AESR2PDE2A
SCHEMBL13838866 0.78 KDM1A (0.61) HTR2APOLQKDM1AHTR2CPDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102803210-A Azetidinyl diamides as monoacylglycerol lipase inhibitors JANSSEN PHARMACEUTICA NV 2012-11-28 CN claimed
EP-3577112-B1 ARYL HYDROCARBON RECEPTOR (AHR) MODULATOR COMPOUNDS PHENEX PHARMACEUTICALS AG (DE) 2020-12-30 EP disclosed
EP-3577115-B1 ARYL HYDROCARBON RECEPTOR (AHR) MODULATOR COMPOUNDS PHENEX PHARMACEUTICALS AG (DE) 2020-12-02 EP disclosed
CN-102803210-A Azetidinyl diamides as monoacylglycerol lipase inhibitors JANSSEN PHARMACEUTICA NV 2012-11-28 CN disclosed
WO-2010088574-A1 AZABENZIMIDAZOLES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2010-08-05 WO disclosed