SCHEMBL13257592

SCHEMBL13257592

Nc1cc(-c2nc(-c3cc(CO)ccc3Cl)c(-c3ncc[nH]3)s2)ccn1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 3/20 0.38
DBF4 Q9UBU7 3/20 0.38
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
PIK3C3 Q8NEB9 1/20 0.33
DYRK1A Q13627 3/20 0.33
KRAS P01116 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
ROCK1 Q13464 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13257053 0.90 PIM1 (0.34) CDC7DBF4PIM1PIM3PIM2
SCHEMBL6842848 0.83 PIK3C3 (0.39) CDC7DBF4PIK3C3MAPK14
SCHEMBL6842852 0.81 CDC7 (0.43) CDC7DBF4PIM1PIM3PIM2
SCHEMBL16938035 0.81 CDC7 (0.42) CDC7DBF4PIM1PIM3PIM2
SCHEMBL16938030 0.76 MAPK14 (0.34) CDC7DBF4MAPK14
SCHEMBL16937936 0.76 CDC7 (0.49) CDC7DBF4PIM1PIM3PIM2
SCHEMBL16938036 0.76 MAPK14 (0.42) CDC7DBF4PIK3C3MAPK14
SCHEMBL6842826 0.76 MAPK14 (0.33) MAPK14
SCHEMBL6842830 0.72 PIK3C3 (0.42) CDC7DBF4PIK3C3MAPK14
SCHEMBL16938031 0.71 MAPK14 (0.43) CDC7DBF4PIK3C3MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010090716-A1 HETEROARYLS AND THEIR USE AS PI3K INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2010-08-12 WO disclosed