SCHEMBL13258024

SCHEMBL13258024

COc1ccc2c(c1)C=C(c1c(C(=O)N3C=C4CC3CN4C)c(C(F)(F)F)nn1C)Cn1c-2c(C2CCCCC2)c2ccc(C(=O)NS(=O)(=O)C(C)C)cc21

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.48
NR1I2 O75469 10/20 0.41
CYP3A4 P08684 3/20 0.40
SCN5A Q14524 2/20 0.40
SCN9A Q15858 3/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL862786 0.90 KCNH2 (0.52) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL862809 0.89 KCNH2 (0.58) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL863120 0.89 KCNH2 (0.51) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL862895 0.89 KCNH2 (0.51) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL863127 0.89 KCNH2 (0.49) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL862782 0.89 KCNH2 (0.49) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL862900 0.88 KCNH2 (0.49) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL863024 0.88 KCNH2 (0.48) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL862896 0.88 KCNH2 (0.48) KCNH2NR1I2CYP3A4SCN5ASCN9A
SCHEMBL863008 0.87 NR1I2 (0.49) KCNH2NR1I2CYP3A4SCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183252-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2015-01-14 EP disclosed
WO-2010093359-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-08-19 WO disclosed
WO-2009029384-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2009-03-05 WO disclosed