SCHEMBL13259017

SCHEMBL13259017

CC1Oc2ccc(Cc3nnc(OCc4c(F)cccc4Cl)n3-c3ccc(F)cc3)cc2O1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 8/20 0.43
KMT2A Q03164 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
HSD11B1 P28845 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13259966 0.84 GPBAR1 (0.59) GPBAR1MAPTHTTHSD11B1ALDH1A1
SCHEMBL10229734 0.82 GPBAR1 (0.64) GPBAR1KMT2AALDH1A1
SCHEMBL13259018 0.79 GPBAR1 (0.67) GPBAR1KMT2AMAPTHTTALDH1A1
SCHEMBL13259961 0.76 GPBAR1 (0.47) GPBAR1KMT2AMAPTHTTHSD11B1
SCHEMBL13259977 0.72 GPBAR1 (0.47) GPBAR1KMT2AMAPTHTTALDH1A1
SCHEMBL13259058 0.69 GPBAR1 (0.52) GPBAR1ALDH1A1
SCHEMBL13259015 0.68 GPBAR1 (0.46) GPBAR1KMT2AMAPTHTTALDH1A1
SCHEMBL13259019 0.67 GPBAR1 (0.47) GPBAR1KMT2AMAPTHTTALDH1A1
SCHEMBL13259965 0.67 GPBAR1 (0.54) GPBAR1ALDH1A1
SCHEMBL10229657 0.67 GPBAR1 (0.66) GPBAR1KMT2AMAPTHTTHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093845-A1 TRIAZOLE AND IMIDAZOLE DERIVATIVES FOR USE AS TGR5 AGONISTS IN THE TREATMENT OF DIABETES AND OBESITY EXELIXIS, INC. (US) 2010-08-19 WO disclosed