SCHEMBL13282973

SCHEMBL13282973

CN(C)S(=O)(=O)N(CCO)Cc1nc(C2CN(CC3CCOCC3)c3c(Cl)cccc32)no1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 18/20 0.46
KCNH2 Q12809 9/20 0.38
CNR2 P34972 3/20 0.38
CYP1A1 P04798 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13282892 0.82 CNR1 (0.57) CNR1KCNH2CNR2NPC1LMNA
SCHEMBL13282843 0.81 CNR1 (0.45) CNR1KCNH2CNR2
SCHEMBL13282974 0.78 CNR1 (0.59) CNR1KCNH2CNR2CYP1A1CYP2C8
SCHEMBL13255242 0.75 CNR1 (0.80) CNR1KCNH2CNR2CYP1A1CYP2C8
SCHEMBL13437810 0.72 CNR1 (0.48) CNR1KCNH2CYP1A1CYP2C8CYP2D6
SCHEMBL13437892 0.70 CNR1 (0.60) CNR1KCNH2CYP1A1CYP2C8CYP2D6
SCHEMBL13437706 0.70 CNR1 (0.60) CNR1KCNH2CYP1A1CYP2C8CYP2D6
SCHEMBL13283075 0.70 CNR1 (0.60) CNR1KCNH2CNR2CYP1A1CYP2C8
SCHEMBL13437780 0.65 CNR1 (0.59) CNR1KCNH2CYP1A1CYP2C8CYP2D6
SCHEMBL13437808 0.64 CNR1 (0.53) CNR1KCNH2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7763732-B2 7-Chloro-3-({5-[N-(morpholin-1-ylcarboxamido)methyl]aminomethyl}-([1,2,4]-thiadiazol-3-yl))-1-(tetrahydropyran-4-yl)methyl-1H-indole, hydrochloride salt; treatment of pain N.V. ORGANON (NL) 2010-07-27 US disclosed