SCHEMBL13286290

SCHEMBL13286290

COc1ccc2nccc(OCC3CCC(NCc4ccc5c(c4)OCCO5)CC3)c2c1

nearest known ligand 0.75

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 15/20 0.75
SLC2A1 P11166 1/20 0.56
MCHR1 Q99705 1/20 0.49
PDE5A O76074 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14514817 1.00 KCNH2 (0.75) KCNH2SLC2A1MCHR1PDE5A
SCHEMBL10226462 1.00 KCNH2 (0.75) KCNH2SLC2A1MCHR1PDE5A
SCHEMBL3694124 1.00 KCNH2 (0.75) KCNH2SLC2A1MCHR1PDE5A
SCHEMBL3126601 0.87 KCNH2 (0.67) KCNH2SLC2A1MCHR1PDE5A
SCHEMBL5263322 0.84 KCNH2 (0.71) KCNH2SLC2A1MCHR1PDE5A
SCHEMBL5263317 0.84 KCNH2 (0.71) KCNH2SLC2A1MCHR1PDE5A
SCHEMBL14341171 0.84 KCNH2 (0.77) KCNH2SLC2A1MCHR1
SCHEMBL5261655 0.84 KCNH2 (0.77) KCNH2SLC2A1MCHR1
SCHEMBL5261660 0.84 KCNH2 (0.77) KCNH2SLC2A1MCHR1
SCHEMBL3683660 0.83 KCNH2 (0.58) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010084152-A1 NOVEL BICYCLIC ANTIBIOTICS BASILEA PHARMACEUTICA AG (CH) 2010-07-29 WO disclosed
US-7223776-B2 Compounds with anti-bacterial activity MORPHOCHEM AG (DE) 2007-05-29 US disclosed
US-7223776-B2 Compounds with anti-bacterial activity MORPHOCHEM AG (DE) 2007-05-29 US disclosed