SCHEMBL13293133

SCHEMBL13293133

C=C(C)c1ccc(Nc2ncnc3c2CN(c2ncccc2Cl)CC3)cc1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 18/20 0.61
P2RX3 P56373 1/20 0.41
PIK3CD O00329 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12973519 0.89 TRPV1 (0.66) TRPV1P2RX3PIK3CD
SCHEMBL13293187 0.87 TRPV1 (0.66) TRPV1
SCHEMBL2845333 0.86 TRPV1 (0.67) TRPV1P2RX3PIK3CD
SCHEMBL2843997 0.85 TRPV1 (0.69) TRPV1
SCHEMBL2851097 0.85 TRPV1 (0.71) TRPV1
SCHEMBL2854722 0.83 TRPV1 (0.87) TRPV1
SCHEMBL14350786 0.81 TRPV1 (0.53) TRPV1
SCHEMBL2850967 0.80 TRPV1 (0.60) TRPV1
SCHEMBL2848814 0.80 TRPV1 (0.62) TRPV1
SCHEMBL12994735 0.80 TRPV1 (0.51) TRPV1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745451-B2 2,3-Difluoro-benzyl)-[6-(5-methyl-pyridin-2-yl)-5,6,7,8-tetrahydro-pyrido[4,3-d]pyrimidin-4-yl]-amine, useful for the prevention and treatment of pain, inflammation, cognitive disorders, anxiety and depression in humans RENOVIS, INC. (US) 2010-06-29 US disclosed