SCHEMBL13293255

SCHEMBL13293255

CNC(=O)N[C@@H](C(=O)N1CCC[C@H]1c1ncc(-c2ccc(C#Cc3ccc(-c4cnc([C@@H]5CCCN5C(=O)CNC(=O)C5CC5)[nH]4)cc3)cc2)[nH]1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.49
PRCP P42785 10/20 0.46
CYP3A4 P08684 3/20 0.45
CYP2C9 P11712 3/20 0.45
NR1I2 O75469 1/20 0.45
ABCB11 O95342 1/20 0.45
OPRK1 P41145 1/20 0.45
CYP1A2 P05177 2/20 0.43
OPRM1 P35372 2/20 0.42
OPRD1 P41143 2/20 0.42
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10145519 0.92 KCNH2 (0.50) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL10145018 0.91 KCNH2 (0.54) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL10144803 0.87 KCNH2 (0.52) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL1747510 0.85 CYP3A4 (0.60) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL1747513 0.85 CYP3A4 (0.60) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL13293096 0.84 KCNH2 (0.50) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL10145208 0.84 CYP3A4 (0.59) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL10144910 0.83 KCNH2 (0.49) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL10145005 0.83 KCNH2 (0.55) KCNH2PRCPCYP3A4CYP2C9NR1I2
SCHEMBL10176641 0.83 KCNH2 (0.49) KCNH2PRCPCYP3A4CYP2C9NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065668-A1 INHIBITORS OF HCV NS5A PRESIDIO PHARMACEUTICALS, INC. (US) 2010-06-10 WO disclosed