SCHEMBL13329451

SCHEMBL13329451

O=C(C1CCCN(c2c3c(nc4ccnn24)CNCC3)C1)N1CCC(C2CCCCC2)CC1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 16/20 0.55
HTR2A P28223 15/20 0.55
HTR2B P41595 15/20 0.55
DGAT2 Q96PD7 3/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14700092 0.96 HTR2C (0.61) HTR2CHTR2AHTR2BDGAT2
SCHEMBL10216996 0.96 HTR2C (0.61) HTR2CHTR2AHTR2BDGAT2
SCHEMBL10216973 0.89 HTR2C (0.67) HTR2CHTR2AHTR2BDGAT2
SCHEMBL10217017 0.89 HTR2C (0.67) HTR2CHTR2AHTR2BDGAT2
SCHEMBL10217911 0.89 HTR2C (0.61) HTR2CHTR2AHTR2BALDH1A1
SCHEMBL13328257 0.88 HTR2C (0.54) HTR2CHTR2AHTR2BDGAT2ALDH1A1
SCHEMBL10218106 0.85 HTR2C (0.59) HTR2CHTR2AHTR2B
SCHEMBL14700109 0.85 HTR2C (0.59) HTR2CHTR2AHTR2B
SCHEMBL10218114 0.85 HTR2C (0.59) HTR2CHTR2AHTR2B
SCHEMBL10219403 0.85 HTR2C (0.62) HTR2CHTR2AHTR2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010060952-A1 6,7,8,9-TETRAHYDRO-5H-1,4,7,10A-TETRAAZA-CYCLOHEPT[F]INDENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS, THEIR USE AND PROCESSES FOR PREPARING THEM BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-03 WO disclosed