SCHEMBL13330593

SCHEMBL13330593

CC(CO)Oc1cc(Cl)c(-c2nnc(-c3cn4cc(C(C)(F)F)cc(Cl)c4n3)s2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.44
NPC1 O15118 4/20 0.35
NFKB1 P19838 4/20 0.35
RAB9A P51151 4/20 0.35
NFKB2 Q00653 4/20 0.35
RELA Q04206 4/20 0.35
SMN1; SMN2 Q16637 4/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
RECQL P46063 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 2/20 0.34
S1PR3 Q99500 2/20 0.33
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3340725 0.94 S1PR1 (0.44) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL13330595 0.88 S1PR1 (0.47) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL3343448 0.87 NPC1 (0.43) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL13331093 0.86 S1PR1 (0.37) S1PR1
SCHEMBL13330599 0.86 NPC1 (0.44) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL13330837 0.85 S1PR1 (0.47) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL13330597 0.84 S1PR1 (0.45) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL13330602 0.82 S1PR1 (0.38) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL3340383 0.82 NPC1 (0.42) S1PR1NPC1NFKB1RAB9ANFKB2
SCHEMBL3340133 0.81 S1PR1 (0.46) S1PR1NPC1NFKB1RAB9ANFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065760-A1 IMIDAZO [1,2A] PYRIDINE DERIVATIVES, THEIR USE AS S1P1 AGONISTS AND METHODS FOR THEIR PRODUCTION EXELIXIS, INC. (US) 2010-06-10 WO disclosed