SCHEMBL13330767

SCHEMBL13330767

Cc1cc(C2CN2)c2nc(-c3nc(-c4cc(F)c(CCC(=O)OC(C)(C)C)cc4Cl)no3)cn2c1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 5/20 0.34
S1PR5 Q9H228 1/20 0.33
CNR2 P34972 2/20 0.32
CNR1 P21554 1/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
KIT P10721 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13331097 0.90 S1PR1 (0.34) S1PR1S1PR5
SCHEMBL3343532 0.85 CNR2 (0.34) S1PR1S1PR5CNR2CNR1
SCHEMBL3342731 0.82 CNR2 (0.33) S1PR1S1PR5CNR2CNR1
SCHEMBL13330803 0.82 CNR2 (0.33) S1PR1CNR2CNR1
SCHEMBL13303833 0.82 SMN1; SMN2 (0.39) S1PR1CNR2CNR1HDAC1HDAC8
SCHEMBL3342478 0.81 S1PR1 (0.37) S1PR1S1PR5CNR2CNR1KIT
SCHEMBL3340738 0.80 S1PR1 (0.37) S1PR1S1PR5CNR2CNR1
SCHEMBL3338104 0.78 S1PR1 (0.38) S1PR1S1PR5
SCHEMBL3340282 0.76 S1PR1 (0.38) S1PR1S1PR5
SCHEMBL3345636 0.75 SMN1; SMN2 (0.40) S1PR1S1PR5CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065760-A1 IMIDAZO [1,2A] PYRIDINE DERIVATIVES, THEIR USE AS S1P1 AGONISTS AND METHODS FOR THEIR PRODUCTION EXELIXIS, INC. (US) 2010-06-10 WO disclosed