SCHEMBL13334753

SCHEMBL13334753

C=CN(/C=N\C)c1ccc(Cn2cc3c(c2N(C)c2ccccc2)c(=O)n(C)c(=O)n3CC(C)C)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 8/20 0.43
PDE1B Q01064 8/20 0.43
PDE1C Q14123 8/20 0.43
PDE2A O00408 5/20 0.43
SLC16A1 P53985 2/20 0.36
BRD4 O60885 1/20 0.34
MAPT P10636 3/20 0.33
TP53 P04637 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 2/20 0.33
LMNA P02545 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
CASP1 P29466 1/20 0.31
HTT P42858 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9608339 0.81 PDE1A (0.48) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL2455867 0.78 PDE1A (0.49) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL2461101 0.77 PDE1A (0.50) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL9608351 0.68 PDE1A (0.44) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL9608334 0.65 PDE1B (0.52) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL2462419 0.65 PDE1A (0.46) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL2453873 0.65 PDE1A (0.48) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL2458000 0.64 PDE1A (0.52) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL9608330 0.64 PDE1A (0.42) PDE1APDE1BPDE1CPDE2ASLC16A1
SCHEMBL2461370 0.63 PDE1A (0.49) PDE1APDE1BPDE1CPDE2ASLC16A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065147-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES, INC. (US) 2010-06-10 WO disclosed