SCHEMBL1334640

SCHEMBL1334640

C=C/C=[C]/CC=CC

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9544944 0.71
SCHEMBL28540176 0.71
SCHEMBL835439 0.67
SCHEMBL7185480 0.67
SCHEMBL122477 0.67
SCHEMBL835095 0.65
SCHEMBL835096 0.65
SCHEMBL5461149 0.65
SCHEMBL16004799 0.65
SCHEMBL28454816 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230241243-A1 CARRIER PARTICLE-DRUG CONJUGATES, SELF-IMMOLATIVE LINKERS, AND USES THEREOF ELUCIDA ONCOLOGY, INC. 2023-08-03 US disclosed
US-9994534-B2 Pain-relieving compositions and uses therefor THE UNIVERSITY OF QUEENSLAND (AU) 2018-06-12 US disclosed
US-20180111910-A1 PAIN-RELIEVING COMPOSITIONS AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2018-04-26 US disclosed
EP-2307013-B1 PAIN-RELIEVING COMPOSITIONS OF FUROXAN NO DONORS AND USES THEREOF UNIV QUEENSLAND (AU) 2016-02-24 EP disclosed
US-20150051404-A1 PAIN-RELIEVING COMPOSITIONS AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2015-02-19 US disclosed
US-8822509-B2 Pain-relieving compositions and uses therefor THE UNIVERSITY OF QUEENSLAND (AU) 2014-09-02 US disclosed
US-20110274713-A1 ANTIGEN-PRESENTING SCAFFOLDS THE UNIVERSITY OF QUEENSLAND (AU) 2011-11-10 US disclosed
EP-2367567-A1 ANTIGEN-PRESENTING SCAFFOLDS The University Of Queensland (AU) 2011-09-28 EP disclosed
US-20110172126-A1 LIBRARIES OF PEPTIDE CONJUGATES AND METHODS FOR MAKING THEM XENOME LTD (AU) 2011-07-14 US disclosed
EP-2331561-A1 LIBRARIES OF PEPTIDE CONJUGATES AND METHODS FOR MAKING THEM Xenome Ltd (AU) 2011-06-15 EP disclosed
EP-2307013-A1 PAIN-RELIEVING COMPOSITIONS OF FUROXAN NO DONORS AND USES THEREOF The University Of Queensland (AU) 2011-04-13 EP disclosed
WO-2010025510-A1 LIBRARIES OF PEPTIDE CONJUGATES AND METHODS FOR MAKING THEM XENOME LTD (AU) 2010-03-11 WO disclosed
WO-2010015022-A1 ANTIGEN-PRESENTING SCAFFOLDS THE UNIVERSITY OF QUEENSLAND (AU) 2010-02-11 WO disclosed
WO-2010000019-A1 PAIN-RELIEVING COMPOSITIONS OF FUROXAN NO DONORS AND USES THEREOF THE UNIVERSITY OF QUEENSLAND (AU) 2010-01-07 WO disclosed
US-20090326017-A1 PAIN-RELIEVING COMPOSITIONS AND USES THEREFOR THE UNIVERSITY OF QUEENSLAND (AU) 2009-12-31 US disclosed
US-6015789-A LUTEINIZING HORMONE RELEASING HORMONE AGONIST AND A LUTEINIZING HORMONE RELEASING HORMONE ANTAGONIST IN COMBINATION, TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2000-01-18 US disclosed
US-5977132-A GALACTORRHEA, HYPERPROLACTINEMIC OVULATION, PROLACTINOMA AND BRAIN TUMORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-11-02 US disclosed
EP-0906115-A1 COMBINED USE OF GnRH AGONIST AND ANTAGONIST Takeda Chemical Industries, Ltd. (JP) 1999-04-07 EP disclosed
WO-1997040846-A1 COMBINED USE OF GnRH AGONIST AND ANTAGONIST TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-11-06 WO disclosed
EP-0781774-A2 Prolactin production inhibitory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-02 EP disclosed