SCHEMBL13354871

SCHEMBL13354871

CNc1n[nH]c2cc(-c3cc(N4C[C@@H](C(=O)NCc5ccc(C)cc5)CC[C@H]4C)nc(N)n3)ccc12

nearest known ligand 0.61

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 20/20 0.61
AURKB Q96GD4 17/20 0.61
ROCK1 Q13464 12/20 0.61
AURKA O14965 11/20 0.61
TGFBR1 P36897 2/20 0.61
PIK3CG P48736 1/20 0.55
PDK1 Q15118 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13354769 0.94 PDPK1 (0.68) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL1319090 0.93 PDPK1 (0.71) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL1321262 0.86 PDPK1 (0.70) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL1318522 0.86 PDPK1 (0.70) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL1318704 0.86 PDPK1 (0.79) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL1320516 0.85 PDPK1 (0.68) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL12122710 0.82 PDPK1 (0.49) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL13354779 0.81 PDPK1 (0.69) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL1318420 0.81 PDPK1 (0.69) PDPK1AURKBROCK1AURKATGFBR1
SCHEMBL1318996 0.81 PDPK1 (0.80) PDPK1AURKBROCK1AURKATGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059658-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-05-27 WO disclosed