SCHEMBL13354872

SCHEMBL13354872

CNc1n[nH]c2cc(-c3cc(N4CCC[C@H](C(=O)Nc5ccccc5)C4)nc(N)n3)ccc12

nearest known ligand 0.84

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 19/20 0.84
AURKB Q96GD4 15/20 0.84
AURKA O14965 11/20 0.84
ROCK1 Q13464 10/20 0.84
TGFBR1 P36897 1/20 0.64
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1317520 0.91 PDPK1 (1.00) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1319787 0.91 PDPK1 (1.00) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1319260 0.86 PDPK1 (0.91) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1319538 0.85 PDPK1 (0.85) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL16966498 0.85 PDPK1 (0.84) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1318359 0.85 PDPK1 (0.84) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1319921 0.84 PDPK1 (0.85) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1319259 0.84 PDPK1 (0.85) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1317749 0.83 PDPK1 (0.81) PDPK1AURKBAURKAROCK1TGFBR1
SCHEMBL1319810 0.83 PDPK1 (0.84) PDPK1AURKBAURKAROCK1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059658-A1 CHEMICAL COMPOUNDS GLAXOSMITHKLINE LLC (US) 2010-05-27 WO disclosed