SCHEMBL13368243

SCHEMBL13368243

CCNC1([C@@H]2CCN(c3c(F)cc4c(=O)c(C=O)cn([C@@H]5C[C@@H]5F)c4c3C#N)C2)CC1

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.36
CYP3A4 P08684 1/20 0.33
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13341781 0.90 KCNH2 (0.39) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL3559878 0.87 KCNH2 (0.49) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL3559880 0.87 KCNH2 (0.49) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL13341780 0.82 KCNH2 (0.36) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL3556609 0.79 CYP3A4 (0.47) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL3556611 0.79 CYP3A4 (0.47) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL13341777 0.77 KCNH2 (0.48) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL13341768 0.76 STAT3 (0.42) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL14014256 0.76 STAT3 (0.42) KCNH2CYP3A4ALDH1A1POLBCHRM2
SCHEMBL14014253 0.75 CYP3A4 (0.45) KCNH2CYP3A4ALDH1A1POLBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7723524-B2 8-cyanoquinolonecarboxylic acid derivative DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2010-05-25 US disclosed