SCHEMBL13399

SCHEMBL13399

CNC(=O)CCc1ccc2cnn(C)c2c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCNC P24863 5/20 0.51
CDK8 P49336 5/20 0.51
ACSS2 Q9NR19 1/20 0.47
CACNA1H O95180 7/20 0.44
HTR2A P28223 1/20 0.42
PASK Q96RG2 1/20 0.42
CDK19 Q9BWU1 1/20 0.42
VNN1 O95497 1/20 0.42
PDE1C Q14123 1/20 0.42
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
MPO P05164 1/20 0.41
KDM2B Q8NHM5 1/20 0.41
KDM4C Q9H3R0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22311425 0.76 CACNA1H (0.58) CCNCCDK8CACNA1HHTR2APASK
SCHEMBL13548299 0.76 CTNNB1 (0.47) CCNCCDK8CACNA1HVNN1PDE1C
SCHEMBL17316406 0.75 KDM4E (0.53) CCNCCDK8CACNA1HVNN1KDM2B
SCHEMBL14800197 0.74 NOTUM (0.52) CCNCCDK8CACNA1HHTR2APASK
SCHEMBL30903411 0.74 NOTUM (0.52) CCNCCDK8CACNA1HHTR2APASK
SCHEMBL30006720 0.74 PDE1C (0.48) CCNCCDK8CACNA1HVNN1PDE1C
SCHEMBL29698372 0.74 CCNC (0.65) CCNCCDK8ACSS2HTR2APASK
SCHEMBL6172461 0.73 HDAC1 (0.57) CCNCCDK8HSD17B1HSD17B2
SCHEMBL14387746 0.73 HDAC1 (0.53) HSD17B1HSD17B2
SCHEMBL20652664 0.72 NPY5R (0.48) CCNCCDK8ACSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011044187-A1 IMINOTHIADIAZINE DIOXIDE COMPOUNDS AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE SCHERING CORPORATION (US) 2011-04-14 WO disclosed