SCHEMBL13403449

SCHEMBL13403449

Nc1cccc(NC(=O)NCCN2CCCCC2)n1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.59
KMT2A Q03164 5/20 0.59
POLB P06746 2/20 0.59
CNR1 P21554 1/20 0.51
KDM4E B2RXH2 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PRMT3 O60678 1/20 0.47
HTR3A P46098 1/20 0.46
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13403450 0.88 SMN1; SMN2 (0.55) KMT2ACNR1KDM4E
SCHEMBL10921358 0.74 KMT2A (1.00) MEN1KMT2APOLBCNR1HTR3A
SCHEMBL10553825 0.74 KMT2A (1.00) MEN1KMT2APOLBCNR1HTR3A
SCHEMBL13403447 0.74 MEN1 (0.51) MEN1KMT2APOLBKDM4E
Bromide SCHEMBL10553700 0.73 KMT2A (0.97) MEN1KMT2APOLBCNR1HTR3A
SCHEMBL14574173 0.73 CNR1 (0.74) MEN1KMT2APOLBCNR1PRMT3
Bromide SCHEMBL10556088 0.73 KMT2A (0.97) MEN1KMT2APOLBCNR1HTR3A
SCHEMBL12974664 0.73 EPHX1 (0.56)
SCHEMBL10923255 0.73 KMT2A (0.97) MEN1KMT2APOLBCNR1HTR3A
SCHEMBL2527623 0.72 MEN1 (0.74) MEN1KMT2APOLBCNR1PRMT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7696217-B2 17-acetamido-4-azasteroid derivatives as androgen receptor modulators MERCK SHARP & DOHME CORP. (US) 2010-04-13 US disclosed
US-7696217-B2 17-acetamido-4-azasteroid derivatives as androgen receptor modulators MERCK SHARP & DOHME CORP. (US) 2010-04-13 US disclosed