SCHEMBL13407693

SCHEMBL13407693

COc1cc(C(=O)NC2CCC[C@H](C[C@@]3(CCC4CCCCC4)NC(=N)N(C)C3=O)C2)cc(Cl)n1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 15/20 0.47
CTSD P07339 13/20 0.47
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
ACKR3 P25106 1/20 0.39
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TSHR P16473 2/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7541925 1.00 BACE1 (0.47) BACE1CTSDTAS1R3TAS1R1TAS1R2
SCHEMBL8197967 0.93 BACE1 (0.51) BACE1CTSDTSHRALDH1A1
SCHEMBL2962292 0.93 BACE1 (0.51) BACE1CTSDTSHRALDH1A1
SCHEMBL13054144 0.93 BACE1 (0.51) BACE1CTSDTSHRALDH1A1
SCHEMBL7554360 0.93 BACE1 (0.51) BACE1CTSDTSHRALDH1A1
SCHEMBL12174286 0.93 BACE1 (0.51) BACE1CTSDTSHRALDH1A1
SCHEMBL12173843 0.93 BACE1 (0.51) BACE1CTSDTSHRALDH1A1
SCHEMBL12500118 0.93 BACE1 (0.48) BACE1CTSDTAS1R3TAS1R1TAS1R2
SCHEMBL13407686 0.90 BACE1 (0.49) BACE1CTSDTSHRALDH1A1
SCHEMBL7541601 0.90 BACE1 (0.49) BACE1CTSDTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7700603-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2010-04-20 US disclosed
US-7700603-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2010-04-20 US disclosed