SCHEMBL1342893

SCHEMBL1342893

CSc1sc(NC(=O)C(=O)Nc2ccc(F)cc2OCC(C)C)nc1CNS(C)(=O)=O

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 8/20 0.36
MYC P01106 2/20 0.35
MAX P61244 2/20 0.35
PTPN1 P18031 1/20 0.33
TRPV1 Q8NER1 5/20 0.33
FBP1 P09467 1/20 0.33
GCK P35557 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2650121 0.95 GCK (0.38) MKNK2MYCMAXPTPN1TRPV1
SCHEMBL1343053 0.92 MKNK2 (0.35) MKNK2TRPV1FBP1GCK
SCHEMBL1342930 0.91 MYC (0.37) MYCMAXPTPN1TRPV1FBP1
SCHEMBL2650118 0.90 GCK (0.33) MKNK2GCK
SCHEMBL1341481 0.90 SLC2A1 (0.36) MYCMAXFBP1
SCHEMBL1342027 0.89 MKNK2 (0.36) MKNK2MYCMAXPTPN1TRPV1
SCHEMBL1342441 0.89 MKNK2 (0.36) MKNK2MYCMAXPTPN1TRPV1
SCHEMBL1343475 0.89 GCK (0.42) MKNK2MYCMAXPTPN1TRPV1
SCHEMBL1343001 0.88 GRM4 (0.37) MKNK2GCK
SCHEMBL1342147 0.87 GCK (0.43) MKNK2MYCMAXPTPN1GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063081-B2 N-(2-Phenoxyphenyl)-N'-(thiazol-2-yl)urea; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-11-22 US disclosed
US-7897628-B2 {2-[3-(4-Methyl-2-[2-methypropoxy]phenyl)-ureido]-thiazol-4-yl}-acetic acid ethyl ester; glucokinase inhibitor; antidiabetic, hypoglycemic agent; activators of glucokinase NOVO NORDISK A/S (DK) 2011-03-01 US disclosed
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents VTV THERAPEUTICS LLC 2004-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040122235-A1 Aryl carbonyl derivatives as therapeutic agents GCK, GCKR, PDK2 MKNK2 469/4885MYC 180/4885MAX 2951/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.