SCHEMBL13459293

SCHEMBL13459293

CNC(=O)c1c(-c2ccc(S)cc2)nn2c(F)cc(-c3cc(C(=O)NC4(c5ccccc5)CC4)ccc3C)cc12

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 6/20 0.53
CYP3A4 P08684 5/20 0.53
KCNH2 Q12809 3/20 0.43
NR1I2 O75469 1/20 0.43
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
F9 P00740 3/20 0.34
TACR3 P29371 1/20 0.34
MAPK14 Q16539 3/20 0.33
TTK P33981 1/20 0.33
DGAT2 Q96PD7 1/20 0.33
PTGER4 P35408 1/20 0.33
AKT1 P31749 1/20 0.33
AKT2 P31751 1/20 0.33
LCK P06239 1/20 0.33
KIT P10721 1/20 0.33
KDR P35968 1/20 0.33
SLC6A9 P48067 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2464955 0.94 CYP2C8 (0.60) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL2464836 0.88 CYP2C8 (0.60) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL13241638 0.85 CYP2C8 (0.59) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL1937126 0.84 CYP2C8 (0.63) CYP2C8CYP3A4KCNH2NR1I2MAPK14
SCHEMBL9911902 0.81 CYP2C8 (0.62) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL667045 0.81 CYP2C8 (0.59) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL2463689 0.80 CYP2C8 (0.46) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL1935064 0.79 CYP2C8 (0.46) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL1934831 0.79 CYP2C8 (0.61) CYP2C8CYP3A4KCNH2NR1I2ROCK2
SCHEMBL1934988 0.78 CYP2C8 (0.57) CYP2C8CYP3A4KCNH2NR1I2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010030538-A2 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2010-03-18 WO disclosed