SCHEMBL13461069

SCHEMBL13461069

N#Cc1cc(-c2cccc(C=O)c2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.49
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
TRIM24 O15164 1/20 0.43
TRIM33 Q9UPN9 1/20 0.43
CDK8 P49336 1/20 0.43
XDH P47989 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
BRD4 O60885 1/20 0.39
DYRK1A Q13627 2/20 0.37
DYRK2 Q92630 2/20 0.37
DYRK1B Q9Y463 2/20 0.37
DYRK3 O43781 1/20 0.37
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL455637 0.81 MYC (0.42) MYCXDHABCG2ALDH1A1NPY5R
SCHEMBL17116812 0.81 MYC (0.54) MYCXDHABCG2USP30NPY5R
SCHEMBL14875772 0.80 CDK8 (0.48) CA12CA1CA2CA9TRIM24
SCHEMBL28166485 0.80 MYC (0.41) MYCXDHABCG2ALDH1A1NPY5R
SCHEMBL9792895 0.79 MYC (0.62) MYCXDHABCG2USP30NPY5R
SCHEMBL31133396 0.79 MYC (0.62) MYCXDHABCG2USP30NPY5R
SCHEMBL16180216 0.79 CDK8 (0.44) CA12CA1CA2CA9TRIM24
SCHEMBL31090305 0.78 MYC (0.58) MYCXDHABCG2ALDH1A1NPY5R
SCHEMBL317097 0.78 MYC (0.58) MYCXDHABCG2ALDH1A1NPY5R
SCHEMBL9792841 0.77 CLK4 (0.61) MYCCLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed