SCHEMBL13467978

SCHEMBL13467978

CCN(c1cccc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)C1CCCCC1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 20/20 0.69
EED O75530 1/20 0.64
RBBP4 Q09028 1/20 0.64
SUZ12 Q15022 1/20 0.64
AEBP2 Q6ZN18 1/20 0.64
EZH1 Q92800 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15710916 0.92 EZH2 (0.77) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL15709792 0.92 EZH2 (0.77) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17804383 0.92 EZH2 (0.65) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL15710369 0.91 EZH2 (0.77) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL15700506 0.90 EZH2 (0.65) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL17148707 0.90 EZH2 (0.65) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL18830035 0.90 EZH2 (0.66) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL13280128 0.90 EZH2 (0.69) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL18829868 0.88 EZH2 (0.75) EZH2EEDRBBP4SUZ12AEBP2
SCHEMBL13468071 0.88 EZH2 (0.75) EZH2EEDRBBP4SUZ12AEBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725314-A1 SUBSTITUTED BENZENE COMPOUNDS Epizyme, Inc. (US) 2020-10-21 EP disclosed
EP-3470396-A1 SUBSTITUTED BENZENE COMPOUNDS Epizyme, Inc. (US) 2019-04-17 EP disclosed
EP-3165520-A1 SUBSTITUTED BENZENE COMPOUNDS Epizyme Inc (US) 2017-05-10 EP disclosed
WO-2012142513-A1 SUBSTITUTED BENZENE COMPOUNDS Epizyme, Inc. (US) 2012-10-18 WO disclosed