SCHEMBL13480258

SCHEMBL13480258

Bc1ccc2c(c1)/C(=C/c1[nH]c3c(c1C)C(=O)N(CCN1CCCC1)CCC3)C(=O)N2

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 18/20 0.75
KDR P35968 18/20 0.75
KIT P10721 11/20 0.75
AURKA O14965 1/20 0.47
AURKB Q96GD4 1/20 0.47
FGFR1 P11362 4/20 0.46
TLK2 Q86UE8 1/20 0.46
SRC P12931 5/20 0.46
LCK P06239 4/20 0.46
FYN P06241 4/20 0.46
YES1 P07947 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13480248 0.99 PDGFRB (0.73) PDGFRBKDRKITAURKAAURKB
SCHEMBL14450418 0.95 PDGFRB (0.80) PDGFRBKDRKITAURKAAURKB
SCHEMBL3136220 0.90 PDGFRB (0.75) PDGFRBKDRKITAURKAAURKB
SCHEMBL3136225 0.90 PDGFRB (0.75) PDGFRBKDRKITAURKAAURKB
SCHEMBL3136212 0.90 PDGFRB (0.75) PDGFRBKDRKITAURKAAURKB
SCHEMBL3133205 0.90 PDGFRB (0.92) PDGFRBKDRKITAURKAFGFR1
SCHEMBL3136234 0.90 PDGFRB (0.75) PDGFRBKDRKITAURKAAURKB
SCHEMBL3133199 0.90 PDGFRB (0.92) PDGFRBKDRKITAURKAFGFR1
SCHEMBL3134399 0.89 PDGFRB (0.73) PDGFRBKDRKITAURKAAURKB
SCHEMBL3135000 0.89 PDGFRB (0.73) PDGFRBKDRKITAURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2157093-A1 PYRROLO-NITROGENOUS HETEROCYCLIC DERIVATIVES, THE PREPARATION AND THE PHARMACEUTICAL USE THEREOF Shanghai Hengrui Pharmaceutical Co. Ltd. (CN) 2010-02-24 EP disclosed