SCHEMBL13480913

SCHEMBL13480913

CSc1nc2ncc(C#N)c(Oc3ccc(Cl)cc3Cl)c2s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 8/20 0.47
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SLC22A12 Q96S37 1/20 0.36
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
ABL1 P00519 1/20 0.35
BCR P11274 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34
SCN9A Q15858 2/20 0.34
S1PR4 O95977 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3193839 0.77 SRC (0.51) SRCABL1BCR
SCHEMBL13481394 0.75 SYK (0.35) SRCSMN1; SMN2
SCHEMBL3189826 0.74 KDR (0.42) SMN1; SMN2NPSR1
SCHEMBL4898811 0.73 SRC (0.56) SRCSLC22A12SLC6A4SLC6A3KCNH2
SCHEMBL3184727 0.73 ACACB (0.37) KCNH2SCN9A
SCHEMBL13480943 0.71 SRC (0.44) SRCABL1BCR
SCHEMBL3192149 0.71 EGFR (0.50) SRCNPSR1MAPT
SCHEMBL3194620 0.71 SRC (0.61) SRCABL1BCR
SCHEMBL13481315 0.70 KDR (0.36)
SCHEMBL3193466 0.69 EGFR (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7659284-B2 Inhibitors of ATP-protein kinase; 7-(3-chloro-4-fluoro-phenylamino)-2-(4-pyrrolidin-1-ylmethyl-phenylamino)-thiazolo[4,5-b]pyridine-6-carbonitrile JANSSEN PHARMACEUTICA NV (BE) 2010-02-09 US disclosed
US-7659284-B2 Inhibitors of ATP-protein kinase; 7-(3-chloro-4-fluoro-phenylamino)-2-(4-pyrrolidin-1-ylmethyl-phenylamino)-thiazolo[4,5-b]pyridine-6-carbonitrile JANSSEN PHARMACEUTICA NV (BE) 2010-02-09 US disclosed