SCHEMBL13499181

SCHEMBL13499181

Cc1ccc(S(=O)(=O)N2C=CNC(=O)[C@H]2CC(=O)NCc2ccc3c(c2)CCC[C@H]3NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.77

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 20/20 0.77
CYP3A4 P08684 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3537951 0.91 BDKRB1 (0.80) BDKRB1CYP3A4
SCHEMBL3530781 0.91 BDKRB1 (0.80) BDKRB1CYP3A4
SCHEMBL3530776 0.91 BDKRB1 (0.80) BDKRB1CYP3A4
SCHEMBL3534907 0.87 BDKRB1 (0.74) BDKRB1
SCHEMBL3535114 0.87 BDKRB1 (0.74) BDKRB1
SCHEMBL3533904 0.87 BDKRB1 (1.00) BDKRB1CYP3A4
SCHEMBL3530949 0.85 BDKRB1 (0.71) BDKRB1
SCHEMBL3530955 0.85 BDKRB1 (0.71) BDKRB1
SCHEMBL3531273 0.85 BDKRB1 (1.00) BDKRB1CYP3A4
SCHEMBL3533329 0.85 BDKRB1 (1.00) BDKRB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7662811-B2 N-(((5R)-5-((1-methylethyl)amino)-5,6,7,8-tetrahydro-2-naphthalenyl)methyl)-2-((2R)-1-((4-methylphenyl)sulfonyl)-3-oxo-1,2,3,4-tetrahydro-2-pyrazinyl)acetamide; for treatment of pain and diseases, such as inflammation mediated diseases AMGEN INC. (US) 2010-02-16 US disclosed