SCHEMBL13501477

SCHEMBL13501477

Cn1cncc1[C@@](N)(c1ccc(Cl)cc1)c1ccc2c(c1)C(c1cccc(Cl)c1)Nc1nnnn1-2

nearest known ligand 0.62

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 17/20 0.62
FNTB P49356 17/20 0.62
PGGT1B P53609 4/20 0.52
CYP3A4 P08684 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13501489 1.00 FNTA (0.62) FNTAFNTBPGGT1BCYP3A4
SCHEMBL3547921 0.95 FNTA (0.58) FNTAFNTBPGGT1BCYP3A4
SCHEMBL1683552 0.89 FNTA (0.49) FNTAFNTBPGGT1B
SCHEMBL3973432 0.84 FNTA (0.44) FNTAFNTB
SCHEMBL13501480 0.84 FNTA (0.44) FNTAFNTBPGGT1B
SCHEMBL3980315 0.83 FNTA (0.43) FNTAFNTB
SCHEMBL13501592 0.81 FNTA (0.59) FNTAFNTBPGGT1BCYP3A4
SCHEMBL13501594 0.81 FNTA (0.59) FNTAFNTBPGGT1BCYP3A4
SCHEMBL7668953 0.80 FNTA (0.42) FNTAFNTBPGGT1B
SCHEMBL13501472 0.80 FNTA (0.55) FNTAFNTBPGGT1BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7655654-B2 Farnesyl transferase inhibiting tricyclic quinazoline derivatives substituted with carbon-linked imidazoles or triazoles JANSSEN PHARMACEUTICA NV (BE) 2010-02-02 US disclosed
US-7511138-B2 Farnesyl transferase inhibiting tricyclic quinazoline derivatives substituted with carbon-linked imidazoles or triazoles JANSSEN PHARMACEUTICA NV (BE) 2009-03-31 US disclosed
US-20080027086-A1 FARNESYL TRANSFERASE INHIBITING TRICYCLIC QUINAZOLINE DERIVATIVES SUBSTITUTED WITH CARBON-LINKED IMIDAZOLES OR TRIAZOLES ANGIBAUD PATRICK R 2008-01-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080027086-A1 FARNESYL TRANSFERASE INHIBITING TRICYCLIC QUINAZOLINE DERIVATIVES SUBSTITUTED WITH CARBON-LINKED IMIDAZOLES OR TRIAZOLES FNTA, FNTB, CYP7A1 FNTA 1/4885FNTB 2/4885PGGT1B 31/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.