SCHEMBL13504792

SCHEMBL13504792

CC1(O)CC(c2nc(-c3ccc(Oc4ccccc4)c(F)c3)c3c(N)nccn23)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TNK2 Q07912 19/20 1.00
IGF1R P08069 1/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359549 1.00 TNK2 (1.00) TNK2IGF1R
SCHEMBL1129603 0.91 TNK2 (1.00) TNK2IGF1R
SCHEMBL1129601 0.91 TNK2 (1.00) TNK2IGF1R
SCHEMBL4361718 0.91 TNK2 (1.00) TNK2IGF1R
SCHEMBL4360605 0.91 TNK2 (1.00) TNK2IGF1R
SCHEMBL4360602 0.91 TNK2 (1.00) TNK2IGF1R
SCHEMBL4361713 0.91 TNK2 (1.00) TNK2IGF1R
SCHEMBL13618371 0.89 TNK2 (0.81) TNK2IGF1R
SCHEMBL13618405 0.88 TNK2 (0.80) TNK2IGF1R
SCHEMBL4358974 0.88 TNK2 (1.00) TNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8481733-B2 Substituted imidazopyr- and imidazotri-azines OSI Pharmaceuticals, LLC (US) 2013-07-09 US claimed
EP-2283020-B1 SUBSTITUTED IMIDAZOPYR-AND IMIDAZOTRI-AZINES OSI PHARM INC (US) 2012-10-31 EP claimed
EP-2283020-B1 SUBSTITUTED IMIDAZOPYR-AND IMIDAZOTRI-AZINES OSI PHARM INC (US) 2012-10-31 EP disclosed