Rufloxacin

Rufloxacin

SCHEMBL135502

CN1CCN(c2c(F)cc3c(=O)c(C(=O)O)cn4c3c2SCC4)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 1.00
ADRA2B P18089 1/20 1.00
MAPK1 P28482 1/20 1.00
ALDH1A1 P00352 5/20 0.98
HPGD P15428 5/20 0.98
HSD17B10 Q99714 4/20 0.98
ALB P02768 1/20 0.55
HRH3 Q9Y5N1 1/20 0.55
TUBB4A P04350 1/20 0.54
POLB P06746 1/20 0.54
TUBB P07437 1/20 0.54
TUBA3C P0DPH7 1/20 0.54
TUBA1B P68363 1/20 0.54
TUBA4A P68366 1/20 0.54
TUBB4B P68371 1/20 0.54
TUBB3 Q13509 1/20 0.54
TUBB2A Q13885 1/20 0.54
TUBB8 Q3ZCM7 1/20 0.54
TUBA3E Q6PEY2 1/20 0.54
TUBA1A Q71U36 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rufloxacin SCHEMBL23282883 0.99 KDM4E (0.98) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL8385662 0.99 KDM4E (1.00) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL8126704 0.99 KDM4E (1.00) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL8390373 0.99 KDM4E (1.00) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL51616 0.99 KDM4E (1.00) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL12505914 0.98 KDM4E (0.98) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL1651162 0.98 KDM4E (0.96) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL574492 0.98 KDM4E (0.98) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL838925 0.98 KDM4E (0.98) KDM4EADRA2BMAPK1ALDH1A1HPGD
Rufloxacin SCHEMBL23581496 0.97 KDM4E (0.96) KDM4EADRA2BMAPK1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4113 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12624057-B2 Bisphosphonate quinolone conjugates and uses thereof BIOVINC, LLC (US) 2026-05-12 US claimed
US-20260090584-A1 SYSTEMS AND METHODS FOR ESTIMATING AEROSOLIZATION EMISSION SCIENTIFIC HORIZONS CONSULTING LLC (US) 2026-04-02 US claimed
EP-4603146-A2 COMBINATION OF ZIDOVUDINE AND FLUOROQUINOLONE ANTIBIOTIC Helperby Therapeutics Limited (GB) 2025-08-20 EP claimed
EP-4590371-A2 SYSTEMS AND METHODS FOR ESTIMATING AEROSOLIZATION EMISSION Scientific Horizons consulting LLC (US) 2025-07-30 EP claimed
EP-4028022-B1 COMBINATION OF ZIDOVUDINE AND FLUOROQUINOLONE ANTIBIOTIC HELPERBY THERAPEUTICS LTD (GB) 2025-07-09 EP claimed
EP-4554627-A1 INHALABLE FORMULATION FOR USE IN THE TREATMENT OF BACTERIAL LUNG INFECTIONS Solmic Biotech GmbH (DE) 2025-05-21 EP claimed
EP-4554939-A1 PCSK9 INHIBITORS AND METHODS OF USE THEREOF Astrazeneca AB (SE) 2025-05-21 EP claimed
US-20250144088-A1 INHALABLE FORMULATION FOR USE IN THE TREATMENT OF BACTERIAL LUNG INFECTIONS Solmic Biotech GmbH (DE) 2025-05-08 US claimed
WO-2025080590-A1 CO-CRYSTALLIZATION OF ACTIVES WITH SACCHARIDE-BASED MOLECULAR FRAMEWORKS SCIENTIFIC HORIZONS CONSULTING LLC (US) 2025-04-17 WO claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
US-5703233-A Quinilone disulfide as intermediates ARCHIMICA SPA (IT) 1997-12-30 US claimed
EP-0725785-B1 PROCESS FOR THE PREPARATION OF RUFLOXACIN AND SALTS THEREOF ARCHIMICA SPA (IT) 1997-07-23 EP claimed
WO-1997024128-A1 OTIC MICROBIAL COMBINATIONS BAYER CORPORATION (US) 1997-07-10 WO claimed
EP-0725785-A1 PROCESS FOR THE PREPARATION OF RUFLOXACIN AND SALTS THEREOF ARCHIMICA SPA (IT) 1996-08-14 EP claimed
US-5532239-A FOR THE TREATMENT OF NEPHROTIC SYNDROMES ASSISTANCE PUBLIQUE - HOPITAUX DE PARIS (FR) 1996-07-02 US claimed
EP-0675880-A1 QUINILONE DISULFIDE AS INTERMEDIATES ARCHIMICA S.P.A. (IT) 1995-10-11 EP claimed
WO-1995011907-A1 PROCESS FOR THE PREPARATION OF RUFLOXACIN AND SALTS THEREOF ARCHIMICA S.P.A. (IT) 1995-05-04 WO claimed
WO-1995011886-A1 QUINILONE DISULFIDE AS INTERMEDIATES ARCHIMICA S.P.A. (IT) 1995-05-04 WO claimed
US-5221741-A Process for the preparation of 9-fluoro-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzothiazine-6-carboxylic acid hydrochloride MEDIOLANUM FARMACEUTICI S.P.A. (IT) 1993-06-22 US claimed
EP-0522277-A1 Process for the preparation of 9-fluoro-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzothiazine-6-carboxylic acid hydrochloride MEDIOLANUM FARMACEUTICI s.r.l. (IT) 1993-01-13 EP claimed