SCHEMBL13560554

SCHEMBL13560554

C=Cc1cc(C#N)cc(Oc2c(Cl)ccc(CN(C(=O)O)C(C)(C)C)c2F)c1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MEP1B Q16820 1/20 0.35
EPAS1 Q99814 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13560574 0.92 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL13560437 0.86 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL13560602 0.85 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL13560541 0.85 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL13560504 0.83 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL13560557 0.81 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19EPAS1
SCHEMBL3017479 0.81 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL5373280 0.80 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL13560474 0.80 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19MEP1BEPAS1
SCHEMBL13560459 0.79 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19MEP1BEPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304419-B2 Chemical compounds GLAXOSMITHKLINE LLC (US) 2012-11-06 US disclosed