SCHEMBL13569822

SCHEMBL13569822

C=C(NC(C)(C)C(F)(F)F)C(C)N1CCC(CNC(=O)c2cc(F)cc(Cl)c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 13/20 0.59
CACNA1H O95180 8/20 0.59
CACNA1G O43497 1/20 0.59
KCNH2 Q12809 11/20 0.56
CYP2D6 P10635 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13569824 0.92 CACNA1I (0.67) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL4274756 0.91 CACNA1I (0.61) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL19113388 0.88 CACNA1I (0.57) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL13569825 0.87 CACNA1H (0.61) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL4271126 0.84 CACNA1I (0.69) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL26082111 0.84 CACNA1I (0.69) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL26082109 0.84 CACNA1I (0.69) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL14770274 0.82 CACNA1I (0.61) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL4274829 0.81 CACNA1I (0.84) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6
SCHEMBL4272441 0.80 CACNA1H (0.63) CACNA1ICACNA1HCACNA1GKCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009146540-A1 N-PIPERIDINYL ACETAMIDE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD (CA) 2009-12-10 WO disclosed