SCHEMBL13575901

SCHEMBL13575901

Cc1ccccc1-c1cnc(N)c(OCC(F)(F)F)n1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATR Q13535 3/20 0.44
PIK3CA P42336 1/20 0.44
PRKDC P78527 1/20 0.44
PDE2A O00408 1/20 0.41
PDE10A Q9Y233 1/20 0.41
ALOX5AP P20292 3/20 0.40
FEN1 P39748 3/20 0.40
SCN9A Q15858 2/20 0.39
SDHB P21912 1/20 0.37
CSF1R P07333 2/20 0.36
HTT P42858 1/20 0.36
HEXA P06865 1/20 0.35
HEXB P07686 1/20 0.35
ADORA2A P29274 1/20 0.35
NUDT1 P36639 1/20 0.35
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
IDO1 P14902 1/20 0.34
METAP2 P50579 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13575849 0.84 ABL1 (0.43) PIK3CAPDE2APDE10AALOX5APFEN1
SCHEMBL10304952 0.83 ATR (0.48) ATRPIK3CAPRKDCALOX5APFEN1
SCHEMBL10305052 0.80 ATR (0.50) ATRPIK3CAPRKDCALOX5APFEN1
SCHEMBL13575848 0.76 ATR (0.44) ATRPRKDCALOX5APFEN1SDHB
SCHEMBL13575846 0.75 PIK3CA (0.41) PIK3CASCN9AADORA2ANUDT1
SCHEMBL28174453 0.75 ATR (0.56) ATRPRKDCALOX5APFEN1HEXA
SCHEMBL13745731 0.72 ADORA2A (0.40) PIK3CAALOX5APFEN1SCN9AADORA2A
SCHEMBL10305022 0.72 HEXA (0.54) ATRPRKDCALOX5APFEN1HEXA
SCHEMBL17204032 0.71 ATR (0.52) ATRPRKDCALOX5APFEN1HEXA
SCHEMBL3134237 0.70 ADORA2A (0.46) PIK3CASCN9AHTTADORA2ANUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090305998-A1 HSP90 INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090305998-A1 HSP90 INHIBITORS HSP90AB1, HSP90AA1, HSP90B1 ATR 2875/4885PIK3CA 645/4885PRKDC 894/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.