SCHEMBL13601224

SCHEMBL13601224

Cc1ccc(Cn2ncc3c(-c4ccco4)nc(N)nc32)cc1

nearest known ligand 0.81

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.81
ADORA1 P30542 17/20 0.81
HDAC1 Q13547 3/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4452013 0.90 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4455442 0.88 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4454421 0.86 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL29051754 0.85 ADORA2A (0.80) ADORA2AADORA1HDAC1
SCHEMBL30514649 0.85 ADORA2A (0.80) ADORA2AADORA1HDAC1
SCHEMBL4447688 0.84 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4452849 0.84 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4459531 0.84 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL4455325 0.83 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4452802 0.83 ADORA2A (1.00) ADORA2AADORA1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629349-B2 Pyrazolo [3,4-d] pyrimidine derivatives and their use as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2009-12-08 US disclosed