SCHEMBL13601248

SCHEMBL13601248

Nc1nc(-c2ccco2)c2cnn(CC(=O)Nc3cccc(Cl)c3)c2n1

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.65
ADORA1 P30542 10/20 0.65
HDAC1 Q13547 10/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4458505 0.89 ADORA2A (0.64) ADORA2AADORA1HDAC1
SCHEMBL4452428 0.87 ADORA2A (0.67) ADORA2AADORA1HDAC1
SCHEMBL4455760 0.86 ADORA2A (0.71) ADORA2AADORA1HDAC1
SCHEMBL4043924 0.84 ADORA2A (0.65) ADORA2AADORA1
SCHEMBL4453241 0.81 ADORA2A (0.61) ADORA2AADORA1HDAC1
SCHEMBL4453263 0.81 ADORA2A (0.65) ADORA2AADORA1HDAC1
SCHEMBL3269889 0.80 ADORA2A (0.65) ADORA2AADORA1
SCHEMBL4452578 0.80 ADORA2A (0.70) ADORA2AADORA1HDAC1
SCHEMBL4452849 0.79 ADORA2A (1.00) ADORA2AADORA1HDAC1
SCHEMBL4457055 0.79 ADORA2A (0.67) ADORA2AADORA1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629349-B2 Pyrazolo [3,4-d] pyrimidine derivatives and their use as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2009-12-08 US disclosed
US-7629349-B2 Pyrazolo [3,4-d] pyrimidine derivatives and their use as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2009-12-08 US disclosed