SCHEMBL13601283

SCHEMBL13601283

Nc1cccc(Cn2ncc3c(-c4nnc[nH]4)nc(N)nc32)c1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.62
ADORA1 P30542 15/20 0.62
ADORA2B P29275 2/20 0.45
ADORA3 P0DMS8 1/20 0.45
HDAC1 Q13547 5/20 0.42
HDAC3 O15379 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MERTK Q12866 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13601277 0.86 ADORA2A (0.66) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL13601270 0.79 ADORA2A (0.71) ADORA2AADORA1ADORA2BADORA3
SCHEMBL4455479 0.79 ADORA2A (0.65) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL4454673 0.78 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL13601285 0.78 ADORA2A (0.65) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL4452802 0.77 ADORA2A (1.00) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL4456600 0.75 ADORA2A (0.66) ADORA2AADORA1ADORA2BADORA3HDAC1
SCHEMBL25548107 0.72 ADORA2A (0.58) ADORA2AADORA1HDAC1MERTK
SCHEMBL24437456 0.70 ADORA2A (0.70) ADORA2AADORA1HDAC1
SCHEMBL4455191 0.67 ADORA2A (0.67) ADORA2AADORA1ADORA2BADORA3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8779078-B2 Method for condensing silyl units using a carbene catalyst BLUESTAR SILICONES FRANCE SAS (FR) 2014-07-15 US disclosed
US-7629349-B2 Pyrazolo [3,4-d] pyrimidine derivatives and their use as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2009-12-08 US disclosed
US-7629349-B2 Pyrazolo [3,4-d] pyrimidine derivatives and their use as purinergic receptor antagonists VERNALIS RESEARCH LIMITED (GB) 2009-12-08 US disclosed