SCHEMBL13601346

SCHEMBL13601346

Cc1cc(C[C@@H](C)C(=O)N2CCN(C3CCN(CC(=O)OCCN(C)C)CC3)CC2)cc2oc(=O)[nH]c12

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 12/20 0.36
CYP3A4 P08684 5/20 0.36
ENPP2 Q13822 1/20 0.33
CALCA P06881 5/20 0.32
RAMP1 O60894 1/20 0.32
CHRM1 P11229 1/20 0.31
BDKRB1 P46663 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13601388 0.98 CALCRL (0.36) CALCRLCYP3A4CALCA
SCHEMBL13601347 0.96 CALCRL (0.35) CALCRLCYP3A4ENPP2CALCARAMP1
SCHEMBL13601389 0.93 CALCRL (0.36) CALCRLCYP3A4CALCA
SCHEMBL13601340 0.92 CALCRL (0.36) CALCRLCYP3A4ENPP2CALCARAMP1
SCHEMBL13601335 0.91 CALCRL (0.37) CALCRLCYP3A4ENPP2CALCACHRM1
SCHEMBL13601342 0.90 CALCRL (0.35) CALCRLCYP3A4ENPP2CALCARAMP1
SCHEMBL13601382 0.90 CALCRL (0.37) CALCRLCYP3A4CALCA
SCHEMBL13601380 0.89 CALCRL (0.38) CALCRLCYP3A4CALCACHRM1
SCHEMBL13601343 0.89 CALCRL (0.35) CALCRLCYP3A4ENPP2CALCA
SCHEMBL13601383 0.89 CALCRL (0.36) CALCRLCYP3A4CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625886-B2 Selected CGRP antagonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-12-01 US disclosed