SCHEMBL13601555

SCHEMBL13601555

CCOC(=O)[C@H]1CCCN1C1CCN(C(=O)[C@H](C)Cc2cc(C)c3[nH]c(=O)oc3c2)CC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 7/20 0.36
CYP3A4 P08684 3/20 0.36
ALDH1A1 P00352 5/20 0.34
KMT2A Q03164 5/20 0.33
MEN1 O00255 4/20 0.33
CALCA P06881 1/20 0.33
EPHX2 P34913 1/20 0.33
SMYD3 Q9H7B4 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
GAA P10253 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13601573 1.00 CALCRL (0.36) CALCRLCYP3A4ALDH1A1KMT2AMEN1
SCHEMBL13601557 0.94 CALCRL (0.35) CALCRLCYP3A4ALDH1A1CALCAEPHX2
SCHEMBL13601574 0.94 CALCRL (0.35) CALCRLCYP3A4ALDH1A1CALCAEPHX2
SCHEMBL13601576 0.93 CALCRL (0.34) CALCRLCYP3A4CALCAEPHX2SMYD3
SCHEMBL13601562 0.93 CALCRL (0.34) CALCRLCYP3A4CALCAEPHX2SMYD3
SCHEMBL13601571 0.92 CALCRL (0.34) CALCRLCYP3A4CALCAEPHX2
SCHEMBL13601585 0.92 CALCRL (0.34) CALCRLCYP3A4CALCAEPHX2
SCHEMBL13601572 0.92 CALCRL (0.33) CALCRLCYP3A4ALDH1A1CALCAEPHX2
SCHEMBL13601563 0.92 CALCRL (0.33) CALCRLCYP3A4EPHX2SMYD3
SCHEMBL13601589 0.92 CALCRL (0.33) CALCRLCYP3A4ALDH1A1CALCAEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7625886-B2 Selected CGRP antagonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-12-01 US disclosed
US-7625886-B2 Selected CGRP antagonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-12-01 US disclosed