SCHEMBL13613646

SCHEMBL13613646

O=C(NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)Nc1cccc2c1CC(O)CC2

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 16/20 0.58
OPRM1 P35372 1/20 0.58
MTOR P42345 2/20 0.50
CCR2 P41597 1/20 0.46
TACR1 P25103 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13613630 0.93 TRPV1 (0.61) TRPV1OPRM1
SCHEMBL2734769 0.91 TRPV1 (0.56) TRPV1OPRM1
SCHEMBL4341559 0.91 TRPV1 (0.59) TRPV1OPRM1
SCHEMBL4332036 0.91 TRPV1 (0.59) TRPV1OPRM1
SCHEMBL4341421 0.91 TRPV1 (0.59) TRPV1OPRM1
SCHEMBL2734529 0.87 TRPV1 (0.56) TRPV1OPRM1
SCHEMBL4347233 0.84 TRPV1 (0.58) TRPV1OPRM1
SCHEMBL13613606 0.84 TRPV1 (0.59) TRPV1OPRM1
SCHEMBL13613654 0.84 TRPV1 (0.73) TRPV1OPRM1
SCHEMBL5111003 0.84 TRPV1 (0.53) TRPV1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612113-B2 Such as N-[4-chloro-3-(trifluoromethyl)phenyl]-N'-(7-hydroxy-5,6,7,8-tetrahydro-1-naphthalenyl)urea; vanilloid receptor antagonists; for treatment of urge urinary incontinence, overactive bladder, chronic pain, neuropathic pain, postoperative pain, rheumatoid arthritic pain, neuralgia, neuropathies, COPD XENTION LIMITED (GB) 2009-11-03 US disclosed
US-7612113-B2 Such as N-[4-chloro-3-(trifluoromethyl)phenyl]-N'-(7-hydroxy-5,6,7,8-tetrahydro-1-naphthalenyl)urea; vanilloid receptor antagonists; for treatment of urge urinary incontinence, overactive bladder, chronic pain, neuropathic pain, postoperative pain, rheumatoid arthritic pain, neuralgia, neuropathies, COPD XENTION LIMITED (GB) 2009-11-03 US disclosed