SCHEMBL13616273

SCHEMBL13616273

COc1c(C)cnc(CN2C/C(=C\c3ccncc3)C(=O)c3c(Cl)nc(N)nc32)c1C

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.59
HSP90AB1 P08238 18/20 0.59
TRAP1 Q12931 2/20 0.46
HSP90B1 P14625 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1789959 0.92 HSP90AA1 (0.59) HSP90AA1HSP90AB1
SCHEMBL1789965 0.92 HSP90AA1 (0.59) HSP90AA1HSP90AB1
SCHEMBL12614054 0.91 HSP90AA1 (0.56) HSP90AA1HSP90AB1TRAP1
SCHEMBL12614057 0.89 HSP90AA1 (0.57) HSP90AA1HSP90AB1TRAP1
SCHEMBL12614031 0.88 HSP90AA1 (0.64) HSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL1787004 0.86 HSP90AA1 (0.62) HSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL1786998 0.86 HSP90AA1 (0.62) HSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL1058516 0.85 HSP90AA1 (0.63) HSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL1058520 0.85 HSP90AA1 (0.63) HSP90AA1HSP90AB1TRAP1HSP90B1
SCHEMBL12613917 0.85 HSP90AA1 (0.57) HSP90AA1HSP90AB1TRAP1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009139834-A1 BIOACTIVE COMPOUNDS FOR TREATMENT OF CANCER AND NEURODEGENERATIVE DISEASES PONIARD PHARMACEUTICALS, INC. (US) 2009-11-19 WO disclosed