SCHEMBL13618149

SCHEMBL13618149

BCCCN1C(=O)COc2ccc(C)cc21

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.62
HTT P42858 1/20 0.62
POLB P06746 3/20 0.61
TP53 P04637 1/20 0.60
PLK1 P53350 1/20 0.58
THRB P10828 1/20 0.56
GAA P10253 2/20 0.56
MAPT P10636 1/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C19 P33261 1/20 0.53
ALDH1A1 P00352 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13618628 0.88 TSHR (0.64) TSHRHTTPOLBTP53PLK1
SCHEMBL4059758 0.88 TSHR (0.64) TSHRHTTPOLBTP53PLK1
SCHEMBL4102493 0.86 TSHR (0.62) TSHRHTTPOLBTP53PLK1
SCHEMBL1764373 0.86 TSHR (0.62) TSHRHTTPOLBTP53PLK1
SCHEMBL10181988 0.86 TSHR (0.62) TSHRHTTPOLBTP53PLK1
SCHEMBL12052569 0.86 TSHR (0.66) TSHRHTTPOLBTP53PLK1
SCHEMBL10181902 0.85 TSHR (0.64) TSHRHTTPOLBTP53PLK1
SCHEMBL1764374 0.85 TSHR (0.61) TSHRHTTPOLBTP53PLK1
SCHEMBL13091199 0.85 TSHR (0.67) TSHRHTTPOLBTP53PLK1
SCHEMBL89401 0.84 TSHR (0.71) TSHRHTTPOLBTP53PLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833816-B1 SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS NOVARTIS AG (CH) 2009-11-11 EP disclosed