SCHEMBL13620858

SCHEMBL13620858

C=Cc1c(OCCCNC(=O)OC(C)(C)C)ccc(/C=C/CCN=[N+]=[N-])c1/C=C\C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 7/20 0.38
CA2 P00918 7/20 0.38
CA12 O43570 5/20 0.38
CA9 Q16790 5/20 0.38
KDM4E B2RXH2 5/20 0.36
TDP1 Q9NUW8 1/20 0.36
POLB P06746 1/20 0.35
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ADRB2 P07550 1/20 0.32
HTR1A P08908 1/20 0.32
BRD4 O60885 2/20 0.32
MAPT P10636 1/20 0.32
CYP1A1 P04798 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2B6 P20813 1/20 0.31
CYP2C19 P33261 1/20 0.31
CYP3A43 Q9HB55 1/20 0.31
AXL P30530 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13730416 0.82 SCN9A (0.39) CA1CA2CA12CA9KDM4E
SCHEMBL13621102 0.80 CA12 (0.37) CA1CA2CA12CA9KDM4E
SCHEMBL13621101 0.74 SCN9A (0.40) CA1CA2CA12CA9KDM4E
SCHEMBL15036905 0.67 CA12 (0.46) CA1CA2CA12CA9TDP1
SCHEMBL13752093 0.66 TDP1 (0.56) CA1CA2CA12CA9TDP1
SCHEMBL16419765 0.66 CA12 (0.46) CA1CA2CA12CA9TDP1
SCHEMBL15452104 0.65 CA1 (0.45) CA1CA2CA12CA9KDM4E
SCHEMBL18569991 0.65 SCN9A (0.48) CA1CA2CA12CA9KDM4E
SCHEMBL15798200 0.65 TDP1 (0.58) CA1CA2CA12CA9KDM4E
SCHEMBL25756209 0.65 TDP1 (0.48) CA1CA2CA12CA9TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009139948-A1 POLY AROMATIC SODIUM CHANNEL BLOCKERS JOHNSON MICHAEL R (US) 2009-11-19 WO disclosed